研究熱點
01、靶點:AHNAK應用:阿爾茨海默病治療新的靶點來源:Multiscale proteomic modeling reveals protein networks driving Alzheimer
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靶點:RPS27L,應用:畜禽產肉性狀遺傳改良、骨骼肌生長發育精準調控及人類肌肉疾病治療,來源:RPS27L Enhances Myogenesis and Muscl
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FLT1(VEGFR-1):血管生成的雙向調節器與疾病治療新靶點
血管內皮生長因子受體(VEGFR)家族一直是熱門靶點,其中,FLT1(VEGFR-1)以其獨特的“雙向調控”角色脫穎而
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靶點:PARP1,應用:腫瘤治療,來源:NASP modulates histone turnover to drive PARP inhibitor resistance Nature,2025 Sep
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蛋白酪氨酸磷酸酶受體D型(Protein tyrosine phosphatase receptor type D, PTPRD)是蛋白酪氨酸磷酸酶
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靶點:SLC45A4,應用:靶向SLC45A4的鎮痛療法,來源:SLC45A4 is a pain gene encoding a neuronal polyamine transporter Nature
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靶點:AKR1B10,應用:結直腸癌(CRC)肝轉移相關研究,來源:AKR1B10 dictates c-Myc stability to suppress colorectal cancer m
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靶點:IRAK4,應用:相關皮膚炎癥的研究與治療,來源:Discovery of Rigid Linker-Based IRAK4 PROTACs with Improved Metabolic
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靶點:GPR146,應用:高血壓治療,來源:GPR146 Facilitates Blood Pressure Elevation and Vascular Remodeling via PIEZO1 Circ
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靶點:ALKBH1,應用:急性髓性白血病(AML)的治療。來源:ALKBH1 drives tumorigenesis and drug resistance via tRNA decoding
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靶點:TRIM21,應用:食管鱗狀細胞癌(ESCC)的治療。來源:TRIM21-mediated K11-linked ubiquitination of ID1 suppresses tumorigene
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靶點:RIPK4,應用:巴索卡-帕帕斯綜合征BPS的研究,來源:RIPK4-mediated MFN2 degradation drives osteogenesis through
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靶點:STC1,應用:針對吞噬信號通路的聯合治療,來源:Stanniocalcin 1 is a phagocytosis checkpoint driiving tumor immune resi
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PHOSPHO1應用:AMD(年齡相關性黃斑變性)治療來源:PHOSPHO1 suppresses ferroptosis in retinal pigment epithelial cell
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LAG3應用:腫瘤免疫治療,來源:Proximity between LAG-3 and the T cell receptor guides suppression of T cell activation and autoimmunity Cell,2025 Jul 24
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Seizure-related 6 homolog(癲癇相關同源物6,SEZ6)是一種跨膜蛋白,最初因與癲癇相關而被發現。其基因定位于染色體17q21 33
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ROR1是一種跨膜糖蛋白,屬于ROR家族,其結構包含胞外免疫球蛋白樣結構域、富含半胱氨酸結構域(Frizzled 結構域)、Kringle結構域
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01靶點:GPATCH4應用:肝細胞癌(HCC)治療來源:GPATCH4 functions as a regulator of nucleolar R-loops in hepatocellular ca
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白細胞介素2(interleukin-2, IL2)是一種關鍵的免疫調節細胞因子,最初因能促進T細胞增殖而被發現,其在免疫系統平衡中發揮 “雙刃劍” 作用:既能激活效應T細胞(Teff)介導抗腫瘤、抗感染免疫
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靶點:IL13Rα1。應用:治療腸道炎癥和蠕蟲感染。來源:Type 2 cytokines act on enteric sensory neurons to regulate neuropeptide-driven hostdefense Science,2025 May 22
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